1179539-52-6Relevant articles and documents
Discovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors
Sinha, Bhaswati,Cao, Zhengyu,Murray, Thomas F.,Aldrich, Jane V.
supporting information; experimental part, p. 7372 - 7375 (2010/04/30)
A series of potent electrophilic affinity labels (IC50= 0.1-5 nM) containing either a bromoacetamide or isothiocyanate based on the μ opioid receptor (MOR) selective peptide dermorphin were prepared. All four analogues exhibited wash resistant inhibition