120115-93-7Relevant articles and documents
RECEPTOR REGULATOR
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, (2010/02/13)
A compound having a partial structure represented by the formula (A) (wherein ring Xa represents a nitrogen-containing ring and R represents optionally substituted amino) or a salt thereof. The compound or salt is highly effective in regulating neuromedin U receptors and is useful as a preventive/therapeutic agent for hypertension, etc.
A VARIANT OF THE BRUYLANTS REACTION. SYNTHESIS OF 4-HETEROARYL-4-ANILINOPIPERIDINES.
Kudzma, Linas V.,Spencer, H. Kenneth,Severnak, Sherry A.
, p. 6827 - 6830 (2007/10/02)
Imines can be generated in situ from α-aminonitriles and efficiently trapped by a variety of lithiated heterocycles.This variation of the Bruylants reaction has proven to be a general method for the synthesis of α-heteroaryl secondary amines.