1245236-15-0Relevant articles and documents
Synthesis and SAR of azolopyrimidines as potent and selective dipeptidyl peptidase-4 (DPP4) inhibitors for type 2 diabetes
Brigance, Robert P.,Meng, Wei,Fura, Aberra,Harrity, Thomas,Wang, Aiying,Zahler, Robert,Kirby, Mark S.,Hamann, Lawrence G.
scheme or table, p. 4395 - 4398 (2010/09/18)
Several pyrazolo-, triazolo-, and imidazolopyrimidines were synthesized and evaluated as inhibitors of DPP4. Of these three classes of compounds, the imidazolopyrimidines displayed the greatest potency and demonstrated excellent selectivity over the other