1361214-48-3Relevant articles and documents
Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging
Fabio, Karine,Guillon, Christophe,Lacey, Carl J.,Lu, Shi-Fang,Heindel, Ned D.,Ferris, Craig F.,Placzek, Michael,Jones, Graham,Brownstein, Michael J.,Simon, Neal G.
, p. 1337 - 1345 (2012/03/26)
SRX246 is a potent, highly selective human vasopressin V1a antagonist that crosses the blood-brain barrier in rats. CNS penetration makes SRX246 an ideal candidate for potential radiolabeling and use in visualization and characterization of the role of th