1380301-57-4Relevant articles and documents
Asymmetric N-allylation of indoles through the iridium-catalyzed allylic alkylation/oxidation of indolines
Liu, Wen-Bo,Zhang, Xiao,Dai, Li-Xin,You, Shu-Li
, p. 5183 - 5187 (2012/07/03)
Two steps can be better than one: An efficient synthesis of enantioenriched N-allylindoles by a one-pot Ir-catalyzed asymmetric allylic alkylation/oxidation reaction of indolines has been realized. The current method features high regioselectivity and enantioselectivity together with a broad range of indoles with varying electronic properties. The utility of this method was demonstrated by the synthesis of dihydropyrrolo[1,2-a]indole derivatives. Copyright