304011-24-3Relevant articles and documents
A synthesis of 2,3,4,5-tetrahydro-1H-3-benzazepines via Pummerer-type cyclization of N-(2-arylethyl)-N-(2-Phenylsulfinylethyl)formamides
Toda, Jun,Ichikawa, Tsuyoshi,Saitoh, Toshiaki,Horiguchi, Yoshie,Sano, Takehiro
, p. 2009 - 2018 (2007/10/03)
A construction of 2,3,4,5-tetrahydro-1H-3-benzazepine ring system (7) was achieved via Pummerer-type cyclization of N-(2-arylethyl)-N-2-(phenylsulfinylethyl)formamides (6). This route produced the benzazepines (10) and (11) in six steps starting from readily available 2-arylethylamines (2) and 2-chloroethyl phenyl sulfide.