34081-76-0Relevant articles and documents
Cinnamoyl derivatives of 7α-aminomethyl-6,14-endo- ethanotetrahydrothebaine and 7α-aminomethyl-6,14-endo- ethanotetrahydrooripavine and related opioid ligands
Rennison, David,Neal, Adrian P.,Cami-Kobeci, Gerta,Aceto, Mario D.,Martinez-Bermejo, Fernando,Lewis, John W.,Husbands, Stephen M.
, p. 5176 - 5182 (2007)
A new series of ligands has been synthesized where the cinnamoyl group of the 14-cinnamoylamino morphinones has been introduced to the 7α-substituent of the 6,14-bridged oripavine series. In vitro the compounds were mostly low efficacy partial agonists or