422518-00-1Relevant articles and documents
Repurposing human Aurora kinase inhibitors as leads for anti-protozoan drug discovery
Patel, Gautam,Roncal, Norma E.,Lee, Patricia J.,Leed, Susan E.,Erath, Jessey,Rodriguez, Ana,Sciotti, Richard J.,Pollastri, Michael P.
, p. 655 - 658 (2014/05/06)
Hesperadin, an established human Aurora B inhibitor, was tested against cultures of Trypanosoma brucei, Leishmania major, and Plasmodium falciparum, and was identified to be a potent proliferation inhibitor. A series of analogs was designed and tested to