57262-94-9 Usage
Description
Setiptiline, also known by its brand name Tecipul, is a tetracyclic antidepressant that functions as a noradrenergic and specific serotonergic antidepressant (NaSSA). It is a potent antagonist of alpha-receptors, exhibiting greater affinity at alpha1 than alpha2 sites, and also serves as an inhibitor of central serotonin receptors. Setiptiline is a mianserin analog, which is reportedly effective in treating depression while maintaining a favorable side-effect profile.
Uses
Used in Pharmaceutical Industry:
Setiptiline is used as an antidepressant medication for the treatment of depression. It works by modulating the levels of norepinephrine and serotonin in the brain, which are neurotransmitters that play a crucial role in regulating mood. The drug's dual action as a noradrenergic and specific serotonergic antidepressant contributes to its effectiveness in managing depressive symptoms.
Additionally, due to its potent antagonist activity at alpha1-receptors, Setiptiline may also be used in the treatment of other conditions that involve the overstimulation of these receptors, such as anxiety or certain cardiovascular disorders. However, further research and clinical trials would be necessary to confirm its efficacy and safety in these applications.
Originator
Organon (Netherlands)
Check Digit Verification of cas no
The CAS Registry Mumber 57262-94-9 includes 8 digits separated into 3 groups by hyphens. The first part of the number,starting from the left, has 5 digits, 5,7,2,6 and 2 respectively; the second part has 2 digits, 9 and 4 respectively.
Calculate Digit Verification of CAS Registry Number 57262-94:
(7*5)+(6*7)+(5*2)+(4*6)+(3*2)+(2*9)+(1*4)=139
139 % 10 = 9
So 57262-94-9 is a valid CAS Registry Number.
InChI:InChI=1/C19H19N/c1-20-11-10-18-16-8-4-2-6-14(16)12-15-7-3-5-9-17(15)19(18)13-20/h2-9H,10-13H2,1H3
