676348-47-3Relevant articles and documents
AMIDE DERIVATIVES COMPRISING HETEROCYCLOALKYL RING
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Paragraph 0346; 0347; 0350, (2020/05/20)
PROBLEM TO BE SOLVED: To provide compounds or pharmacologically acceptable salts thereof that have excellent EP300 and/or CREBBP histone acetyltransferase inhibitory activity. SOLUTION: The invention provides compounds represented by the formula (1) in the figure or pharmacologically acceptable salts thereof. (In the formula (1), ring Q1, ring Q2, ring Q3, X and L are as defined in the specification.) SELECTED DRAWING: None COPYRIGHT: (C)2020,JPO&INPIT
A mild and general one-pot preparation of cyanoethyl-protected tetrazoles
Kennedy, Lawrence J.
experimental part, p. 2010 - 2013 (2010/06/14)
Described herein is a mild and general one-pot procedure for the conversion of cyanoethyl amides to cyanoethyl-protected tetrazoles with azidotrimethylsilane via the intermediacy of imidoyl chlorides generated in situ with phosphorus pentachloride. This s