894407-00-2Relevant articles and documents
Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-S N2′ reactions and their use in the preparation of low-molecule CXCR4 antagonists
Niida, Ayumu,Tanigaki, Hiroaki,Inokuchi, Eriko,Sasaki, Yoshikazu,Oishi, Shinya,Ohno, Hiroaki,Tamamura, Hirokazu,Wang, Zixuan,Peiper, Stephen C.,Kitaura, Kazuo,Otaka, Akira,Fujii, Nobutaka
, p. 3942 - 3951 (2007/10/03)
Organocopper-mediated anti-SN2′ reactions of γ-phosphoryloxy-α,β-unsaturated-δ-lactams were used to prepare highly functionalized diketopiperazine mimetics. The substrate phosphates 24, 32, and 47 were prepared from a-amino acid-derived allylic