956102-17-3Relevant articles and documents
The discovery and optimisation of benzazepine sulfonamide and sulfones as potent agonists of the motilin receptor
Bailey, James M.,Scott, Jackie S.,Basilla, Jonathan B.,Bolton, Victoria J.,Boyfield, Izzy,Evans, David G.,Fleury, Etienne,Heightman, Tom D.,Jarvie, Emma M.,Lawless, Kirk,Matthews, Kim L.,McKay, Fiona,Mok, Hindy,Muir, Alison,Orlek, Barry S.,Sanger, Gareth J.,Stemp, Geoffrey,Stevens, Alexander J.,Thompson, Mervyn,Ward, John,Vaidya, Kalindi,Westaway, Susan M.
scheme or table, p. 6452 - 6458 (2010/05/02)
Optimisation of a series of benzazepine sulfonamide hit compounds identified from high throughput screening led to the discovery of a new series of tractable, potent motilin receptor agonists.