101536-79-2Relevant articles and documents
Structure Activity Relationships for a Series of Eticlopride-Based Dopamine D2/D3Receptor Bitopic Ligands
Battiti, Francisco O.,Boateng, Comfort A.,Bonifazi, Alessandro,Cao, Jianjing,Chen, Li,Chitsazi, Rezvan,Lee, Kuo Hao,Newman, Amy Hauck,Ravi, Saiprasad,Shaik, Anver Basha,Shi, Lei
, p. 15313 - 15333 (2021/11/01)
The crystal structure of the dopamine D3 receptor (D3R) in complex with eticlopride inspired the design of bitopic ligands that explored (1) N-alkylation of the eticlopride's pyrrolidine ring, (2) shifting of the position of the pyrrolidine nitrogen, (3)
Synthesis and in vitro affinity for dopamine D-2 receptor of N-fluorine-substituted analogs of eticlopride
Fukumura,Dohmoto,Maeda,Fukuzawa,Kojima
, p. 1740 - 1742 (2007/10/02)
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