1027243-08-8Relevant articles and documents
Cyclopropane-derived peptidomimetics. Design, synthesis, evaluation, and structure of novel HIV-1 protease inhibitors
Martin, Stephen F.,Dorsey, Gordon O.,Gane, Todd,Hillier, Michael C.,Kessler, Horst,Baur, Matthias,Math?, Barbara,Erickson, John W.,Bhat, T. Nagarajan,Munshi, Sanjeev,Gulnik, Sergei V.,Topol, Igor A.
, p. 1581 - 1597 (2007/10/03)
Toward establishing the general efficacy of using trisubstituted cyclopropanes as peptide mimics to stabilize extended peptide structures, the cyclopropanes 20a-d were incorporated as replacements into 9-13, which are analogues of the known HIV-1 protease