1056938-94-3Relevant articles and documents
New optically active 4-alkoxyprolinol ethers derived from trans-4-Hydroxy-L-proline
Friedemann, Nora M.,Eustergerling, Astrid,Nubbemeyer, Udo
experimental part, p. 837 - 843 (2012/03/11)
(2S,4R)-trans-4-Hydroxy-L-proline has been used as thechiral-pool source in the efficient syntheses of optically active protected 4-hydroxyprolinols. After N-acyl protection andester formation, the first ether moiety was introduced maintaining the chiral
ADENOSINE DERIVATIVES HAVING A2A RECEPTOR ACTIVITY
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Page/Page column 51-52, (2008/06/13)
Compounds of (I), or stereoisomers or pharmaceutically acceptable salts thereof, where W, R1, R2, R3 and R4 have the meanings as indicated in the specification, are useful for treating conditions mediated by activation of the adenosine A2A receptor, especially inflammatory or obstructive airways diseases. Pharmaceutical compositions that contain the compounds and a process for preparing the compounds are also described.