1058608-67-5Relevant articles and documents
Direct preparation of arylethynylzinc bromides and their application to cross-coupling reactions
Joo, Seong-Ryu,Kim, Jong-Sung,Kim, Seung-Hoi
, p. 3267 - 3270 (2017)
A novel synthetic protocol for the preparation of arylethynylzinc bromides has been developed. Thus-obtained organozinc reagents were successfully employed in the subsequent cross-coupling reactions with a broad range of aryl halides providing the corresponding alkynylated compounds in good to excellent yields.
Synthesis, Optimization, ADME Analysis, and Antioxidant Activity of 2-(Arylethynyl)-3-ethynylthiophenes
Kavak,Algso,Konus,Y?lmaz,Lazo?lu,Karaa?a?,Kivrak
, p. 91 - 99 (2021/03/04)
Abstract: 2,3-Dialkynylthiophene derivatives were synthesized by using regio- andstereocontrolled Pd-catalyzed Sonogashira coupling and desilylation reactions.The synthesized compounds were analyzed in silico for their pharmacokineticparameters, general t
Domino C-N coupling/annulation versus C-N coupling/ hydroamination of 2-alkynyl-3-bromobenzothiophenes and 2-alkynyl-3-bromothiophenes. highly efficient synthesis of benzothieno[3,2-b]quinolines and thieno[3,2-b]pyrroles
Salman, Ghazwan Ali,Hussain, Munawar,Iaroshenko, Viktor,Villinger, Alexander,Langer, Peter
scheme or table, p. 331 - 336 (2011/04/16)
While the palladium-catalyzed reaction of 2-alkynyl-3-bromothiophenes with anilines afforded thienopyrroles by a domino C-N coupling/hydroamination process, the reaction of 2-alkynyl-3-bromobenzothiophenes with anilines resulted, under identical condition