1069123-92-7Relevant articles and documents
Copper(I)-catalyzed, one-pot synthesis of multisubstituted indoles from 2-iodoanilines and ethyl buta-2,3-dienoate
Wang, Xianxue,Liu, Jin,Guo, Han,Ma, Chao,Gao, Xiai,Zhou, Kang,Huang, Guosheng
, p. 1037 - 1042 (2012)
Reactions of 2-iodoanilines with ethyl buta-2,3-dienoate catalyzed by potassium carbonate and CuI in one pot generate the corresponding ethyl 2-methyl-1H-indole-3-carboxylate products in moderate yields under mild conditions. Georg Thieme Verlag Stuttgart · New York.
Copper-catalyzed synthesis of 2,3-disubstituted indoles from ortho-haloanilines and β-keto esters/β-diketone
Liu, Xiao-Guang,Li, Zi-Hao,Xie, Jian-Wei,Liu, Ping,Zhang, Jie,Dai, Bin
supporting information, p. 653 - 657 (2016/01/15)
Tetrazole-1-acetic acid was identified as an efficient ligand to promote copper-catalyzed domino reaction of ortho-iodo/bromo-anilines with β-keto esters/β-diketone for 2,3-disubstituted indoles' synthesis with high yields under mild conditions. The proto