109216-58-2Relevant articles and documents
Synthesis and structure-activity relationships of potent and orally active 5-HT4 receptor antagonists: Indazole and benzimidazolone derivatives
Schaus, John M.,Thompson, Dennis C.,Bloomquist, William E.,Susemichel, Alice D.,Calligaro, David O.,Cohen, Marlene L.
, p. 1943 - 1955 (2007/10/03)
A series of indole-3-carboxamides, indazole-3-carboxamides, and benzimidazolone-3-carboxamides was synthesized and evaluated for antagonist affinity at the 5-HT4 receptor in the rat esophagus. The endo-3-tropanamine derivatives in the indazole
Indazoles as indole bioisosteres: Synthesis and evaluation of the tropanyl ester and amide of indazole-3-carboxylate as antagonists at the serotonin 5HT3 receptor
Fludzinski,Evrard,Bloomquist,Lacefield,Pfeifer,Jones,Deeter,Cohen
, p. 1535 - 1537 (2007/10/02)
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