1094322-44-7Relevant articles and documents
Discovery of selective nonpeptidergic neuropeptide FF2 receptor agonists
Gaubert, Gilles,Bertozzi, Fabio,Kelly, Nicholas M.,Pawlas, Jan,Scully, Audra L.,Nash, Norman R.,Gardell, Luis R.,Lameh, Jelveh,Olsson, Roger
supporting information; experimental part, p. 6511 - 6514 (2010/03/26)
We report the discovery and initial characterization of a novel class of selective NPFF2 agonists. HTS screening using R-SAT, a whole cell based functional assay, identified a class of aryliminoguanidines as NPFF1 and NPFF2 ligands. Subsequent optimizatio