1158974-92-5Relevant articles and documents
Synthesis of boronic acid derivatives of tyropeptin: Proteasome inhibitors
Watanabe, Takumi,Momose, Isao,Abe, Masatoshi,Abe, Hikaru,Sawa, Ryuichi,Umezawa, Yoji,Ikeda, Daishiro,Takahashi, Yoshikazu,Akamatsu, Yuzuru
supporting information; scheme or table, p. 2343 - 2345 (2009/12/07)
Boronic acid derivatives of tyropeptin were synthesized with TP-110 as the lead compound. Due to the lability of the aminoboronic acid moiety, careful design of the deprotection and coupling sequence was required. Liquid-liquid partition chromatography wa