1188931-97-6Relevant articles and documents
Vitamin D receptor agonist/histone deacetylase inhibitor molecular hybrids
Lamblin, Marc,Dabbas, Basel,Spingarn, Russell,Mendoza-Sanchez, Rodrigo,Wang, Tian-Tian,An, Beum-Soo,Huang, Dao Chao,Kremer, Richard,White, John H.,Gleason, James L.
experimental part, p. 4119 - 4137 (2010/08/06)
Incorporation of zinc-binding groups into the side-chain of 1α,25-dihydroxyvitamin D3 (1,25D) fully bifunctional hybrid molecules which act both as vitamin D receptor agonists and histone deacetylase inhibitors. These bifunctional hybrids displ