1258291-80-3

Basic information

• Product Name: (2S,3aS,7aS)-1-[(S)-N-[(S)-1-carboxy-butyl]alanyl]hexahydro-2-indolinecarboxylic acid 1-ethyl ester para-toluenesulfonate
• Synonyms: (2S,3aS,7aS)-1-[(S)-N-[(S)-1-carboxy-butyl]alanyl]hexahydro-2-indolinecarboxylic acid 1-ethyl ester para-toluenesulfonate
• CAS NO: 1258291-80-3
• Molecular Weight: 540.678
• Mol File: 1258291-80-3.mol
• Article Data: 1

Chemical Properties

• CAS DataBase Reference: (2S,3aS,7aS)-1-[(S)-N-[(S)-1-carboxy-butyl]alanyl]hexahydro-2-indolinecarboxylic acid 1-ethyl ester para-toluenesulfonate(CAS DataBase Reference)
• NIST Chemistry Reference: (2S,3aS,7aS)-1-[(S)-N-[(S)-1-carboxy-butyl]alanyl]hexahydro-2-indolinecarboxylic acid 1-ethyl ester para-toluenesulfonate(1258291-80-3)
• EPA Substance Registry System: (2S,3aS,7aS)-1-[(S)-N-[(S)-1-carboxy-butyl]alanyl]hexahydro-2-indolinecarboxylic acid 1-ethyl ester para-toluenesulfonate(1258291-80-3)

Safety Data

• Hazardous Substances Data: 1258291-80-3(Hazardous Substances Data)

Upstream product

• 107133-36-8 perindopril tert-butylamine 
• 104-15-4 toluene-4-sulfonic acid 
• 82834-16-0 Perindopril 

Relevant articles and documents

PERINDOPRIL TOSYLATE

The present invention relates to a novel salt of perindopril, namely the paratoluene sulfonic acid salt. The present invention also relates to an amorphous form of the perindopril paratoluene sulfonic acid salt. The invention further relates to processes for the preparation of the novel salt and the amorphous form thereof. The invention also relates to pharmaceutical compositions comprising the perindopril tosylate for the treatment of hypertension and heart failure.