1261298-37-6Relevant articles and documents
Synthesis and pharmacological characterization of 5-phenyl-2-[2-(1- piperidinylcarbonyl)phenyl]-2,3-dihydro-1H-pyrrolo[1,2-c]imidazol-1-ones: A new class of Neuropeptide S antagonists
Micheli, Fabrizio,Di Fabio, Romano,Giacometti, Angelo,Roth, Adelheid,Moro, Elisa,Merlo, Giancarlo,Paio, Alfredo,Merlo-Pich, Emilio,Tomelleri, Silvia,Tonelli, Federica,Zarantonello, Paola,Zonzini, Laura,Capelli, Anna Maria
, p. 7308 - 7311 (2011/02/21)
A new class of selective NPS antagonist was developed starting from a commercially available product identified by screening activities. Experimental NMR observations and computational experiments allowed the discovery of a new class of derivatives. 5-Phe