1301724-94-6Relevant articles and documents
Selective chemical oxidation of risperidone: A straightforward and cost-effective synthesis of paliperidone
Riva, Renata,Banfi, Luca,Castaldi, Graziano,Ghislieri, Diego,Malpezzi, Luciana,Musumeci, Francesca,Tufaro, Roberto,Rasparini, Marcello
, p. 2319 - 2325 (2011)
A very short and cost-effective synthesis of the commercial drug paliperidone has been achieved starting from its parent compound risperidone, through a thoroughly optimized oxidation with air under basic conditions. A very short and cost-effective synthesis of the commercial drug paliperidone (1) has been achieved starting from its parent compound risperidone, through a thoroughly optimized oxidation with air under basic conditions. Copyright