1310087-47-8Relevant articles and documents
Discovery of pyrimidine carboxamides as potent and selective CCK1 receptor agonists
Wang, Liping,Hubert, James A.,Lee, Susan J.,Pan, Jie,Qian, Su,Reitman, Marc L.,Strack, Alison M.,Weingarth, Drew T.,MacNeil, Douglas J.,Weber, Ann E.,Edmondson, Scott D.
scheme or table, p. 2911 - 2915 (2011/06/24)
A series of six-membered heterocycle carboxamides were synthesized and evaluated as cholecystokinin 1 receptor (CCK1R) agonists. A pyrimidine core proved to be the best heterocycle, and SAR studies resulted in the discovery of analog 5, a potent and struc
