1334763-86-8Relevant articles and documents
Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin- 2-yl)-4-(quinoxalin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
Jin, Cheng Hua,Sreenu, Domalapally,Krishnaiah, Maddeboina,Subrahmanyam, Vura Bala,Rao, Kota Sudhakar,Nagendra Mohan, Annaji Venkata,Park, Chul-Yong,Son, Jee-Yeon,Son, Do-Hyun,Park, Hyun-Ju,Sheen, Yhun Yhong,Kim, Dae-Kee
, p. 3917 - 3925 (2011/11/07)
A series of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl) pyrazoles 14a-d, 15a-d, 17a, 17b, 18a-d, 19a, and 19b has been synthesized and evaluated for their ALK5 inhibitory activity in an enzyme assay and in a cell-based luciferase reporte