1360599-16-1Relevant articles and documents
Palladium-catalyzed direct C2 arylation of N-substituted indoles with 1-aryltriazenes
Liu, Can,Miao, Tao,Zhang, Lei,Li, Pinhua,Zhang, Yicheng,Wang, Lei
, p. 2584 - 2589 (2014/10/15)
A novel and efficient palladium-catalyzed C2 arylation of N-substituted indoles with 1-aryltriazenes for the synthesis of 2-arylindoles was developed. In the presence of BF3?OEt2 and palladium(II) acetate (Pd(OAc)2), N-substituted indoles reacted with 1-aryltriazenes in N,N-dimethylacetamide (DMAC) to afford the corresponding aryl-indole-type products in good to excellent yields.