1436417-01-4Relevant articles and documents
Structure–Activity Relationships of 1-Benzoylazulenes at the OX1 and OX2 Orexin Receptors
Turku, Ainoleena,Leino, Teppo O.,Karhu, Lasse,Yli-Kauhaluoma, Jari,Kukkonen, Jyrki P.,Wallén, Erik A. A.,Xhaard, Henri
, p. 965 - 981 (2019)
We previously demonstrated the potential of di- or trisubstituted azulenes as ligands (potentiators, weak agonists, and antagonists) of the orexin receptors. In this study we investigated 27 1-benzoylazulene derivatives, uncovering seven potentiators of t
Site-Selective Addition of Maleimide to Indole at the C-2 Position: Ru(II)-Catalyzed C-H Activation
Lanke, Veeranjaneyulu,Bettadapur, Kiran R.,Prabhu, Kandikere Ramaiah
supporting information, p. 4662 - 4665 (2015/10/12)
Synthesis of 3-(indol-2-yl)succinimide derivatives is presented using a directing group strategy. Selective functionalization of C-2 in the presence of highly reactive C-3 in indole derivatives has been achieved. A conjugate addition product instead of He