1446021-18-6Relevant articles and documents
Efficient Suzuki-Miyaura mono-arylation of symmetrical diiodo(hetero)arenes
Sapegin, Alexander,Krasavin, Mikhail
, p. 1948 - 1951 (2018)
A reliable protocol for converting 1,4-diiodo-2,3,5,6-tetrafluorobenzene into 1-(hetero)aryl-4-iodo-2,3,5,6-tetrafluorobenzene derivatives has been lacking in the literature. We have identified optimal conditions to achieve this conversion in good yields and have minimized formation of the bis-coupling product. The newly identified protocol involving the use of a syringe pump has been extended to other symmetrical diiodo(hetero)arenes.
AZETIDINE DERIVATIVES
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Paragraph 0554; 0555; 0556; 0557; 0558, (2013/06/28)
Azetidine derivatives of which the following is exemplary and their use in the treatment of obesity, diabetes or dyslipidemia.
NEW AZETIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF
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Page/Page column 77; 78, (2013/07/19)
The invention relates to new azetidine derivatives of the formula (I), to their use as medicaments, to methods for their therapeutic use and to pharmaceutical compositions containing them.