1467063-99-5Relevant articles and documents
Highly regioselective palladium-catalyzed direct cross-coupling of imidazo[1,2-a]pyridines with arylboronic acids
Zhao, Limin,Zhan, Haiying,Liao, Jinqiang,Huang, Jianping,Chen, Qinlin,Qiu, Huifang,Cao, Hua
, p. 65 - 67 (2014/08/18)
A highly regioselective method for the palladium-catalyzed direct cross-coupling of imidazo[1,2-a]pyridines with arylboronic acids has been developed by using O2 as oxidant. This process can be applied to a wide range of imidazo[1,2-a]pyridines and arylboronic acids with excellent C-3-regioselectivity. It provides a new way for developing CC bond-forming processes of multisubstituted imidazo[1,2-a]pyridines, which are common structural motifs in natural products and pharmaceuticals.