1606994-77-7Relevant articles and documents
Tandem Phospha-Michael Addition/N-Acylation/ Intramolecular Wittig Reaction of aza-o-Quinone Methides: Approaches to 2,3-Disubstituted Indoles
Hua, Ting-Bi,Chao, Fei,Wang, Long,Yan, Chen-Yang,Xiao, Cong,Yang, Qing-Qing,Xiao, Wen-Jing
supporting information, p. 2615 - 2619 (2020/05/18)
A tandem phospha-Michael addition/N-acylation/intramolecular Wittig reaction of in situ formed aza-o-QMs is disclosed. This approach features high functional group tolerance and provides a convenient and practical access to biologically significant indole derivatives (37 examples, up to 91% yield) under mild reaction conditions. (Figure presented.).
A robust, well-defined homogeneous silver(I) catalyst for mild intramolecular hydroamination of 2-ethynylanilines leading to indoles
McNulty, James,Keskar, Kunal
, p. 1622 - 1629 (2014/03/21)
A highly efficient, chemically stable and well-defined homogeneous silver(I) catalyst is reported for the room temperature, intramolecular hydroamination of 2-alkynylanilines leading to indole derivatives. Copyright