184951-65-3Relevant articles and documents
5-HT1A-versus D2-receptor selectivity of flesinoxan and analogous N4-substituted N1-arylpiperazines.
Kuipers,Kruse,van Wijngaarden,Standaar,Tulp,Veldman,Spek,IJzerman
, p. 300 - 312 (1997)
We investigated the structural requirements for high 5-HT1A affinity of the agonist flesinoxan and its selectivity versus D2 receptors. For this purpose a series of arylpiperazine congeners of flesinoxan were synthesized and evaluated for their ability to