188822-63-1

Basic information

• Product Name: Phenol, 4-bromo-5-[[[2-(4-hydroxyphenyl)ethyl]methylamino]methyl]-2-methoxy-
• CAS NO: 188822-63-1
• Molecular Formula: C17H20BrNO3
• Molecular Weight: 366.255
• Mol File: 188822-63-1.mol
• Article Data: 4

Chemical Properties

• CAS DataBase Reference: Phenol, 4-bromo-5-[[[2-(4-hydroxyphenyl)ethyl]methylamino]methyl]-2-methoxy-(CAS DataBase Reference)
• NIST Chemistry Reference: Phenol, 4-bromo-5-[[[2-(4-hydroxyphenyl)ethyl]methylamino]methyl]-2-methoxy-(188822-63-1)
• EPA Substance Registry System: Phenol, 4-bromo-5-[[[2-(4-hydroxyphenyl)ethyl]methylamino]methyl]-2-methoxy-(188822-63-1)

Safety Data

• Hazardous Substances Data: 188822-63-1(Hazardous Substances Data)

Usage

General Description

"Phenol, 4-bromo-5-[[[2-(4-hydroxyphenyl)ethyl]methylamino]methyl]-2-methoxy-" is a complex chemical compound containing phenol, bromine, hydroxyphenyl, ethyl, methylamino, and methoxy groups. Phenol, 4-bromo-5-[[[2-(4-hydroxyphenyl)ethyl]methylamino]methyl]-2-methoxy- has potential pharmaceutical applications due to its structural properties, including its bromine substitution which can alter its biological activity. The presence of the hydroxyphenyl and methylamino groups suggest potential antioxidant and medicinal properties, while the methoxy group may contribute to its bioavailability and metabolic stability. Further research and testing may be needed to determine the full range of potential uses for this compound."

Upstream product

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Relevant articles and documents

A concise, scaleable synthesis of narwedine

A concise, scaleable synthesis of narwedine from 3,4- dimethoxybenzaldehyde is described. The procedure features a simple modification to the Barton phenolic coupling route.

Preparation method of galanthamine key intermediate

The invention discloses a preparation method of galanthamine key intermediate -N-methyl(4-leptodactyline)-2-bromo-5-hydroxyl-4-methoxybenzylamine. The preparation method comprises the following steps: by taking 2-bromo-5-benzyloxy-4-methoxybenzaldehyde, benzyloxyphenyl ethanol and methylamine hydrochloride as raw materials, condensing, degrading and performing debenylation reaction to prepare N-methyl(4-leptodactyline)-2-bromo-5-hydroxyl-4-methoxybenzylamine. Cheap and easily available raw materials are adopted in the method, so that the production cost can be effectively controlled, the operation is simple, and the reaction conditions are mild. The intermediate is used for industrial synthesis of galanthamine, and the problem that the yield from the industrial production of galanthamine is low can be effectively solved.