190663-25-3Relevant articles and documents
Triflic anhydride mediated synthesis of 3,4-dihydroquinazolines: A three-component one-pot tandem procedure
Magyar, Christina L.,Wall, Tyler J.,Davies, Steven B.,Campbell, Molly V.,Barna, Haven A.,Smith, Sydney R.,Savich, Christopher J.,Mosey, R. Adam
, p. 7995 - 8000 (2019)
A one-pot three-component tandem reaction involving a key Pictet-Spengler-like annulation step has been developed, providing an efficient method for the synthesis of 3,4-dihydroquinazolines in moderate to good yields from amides, aldehydes, and amines. The multicomponent triflic anhydride mediated reaction tolerates the installation of numerous functional groups, affording extensive diversity about the heterocyclic scaffold.
1-(2-alkanamidoethyl)-6-methoxyindole derivatives: A new class of potent indole melatonin analogues
Tarzia, Giorgio,Diamantini, Giuseppe,Di Giacomo, Barbara,Spadoni, Gilberto,Esposti, Daniele,Nonno, Romolo,Lucini, Valeria,Pannacci, Marilou,Fraschini, Franco,Stankov, Bojidar Michaylov
, p. 2003 - 2010 (2007/10/03)
A new series of indole melatonin analogues, bearing the amido ethyl side chain attached at the N-1 position of the indole nucleus, were synthesized and tested for their affinity for the melatonin receptor isolated from quail optic tecta in a series of in
