198968-77-3Relevant articles and documents
Synthesis and biological properties of new constrained CCK-B antagonists: Discrimination of two affinity states of the CCK-B receptor on transfected CHO cells
Bellier, Bruno,McCort-Tranchepain, Isabelle,Ducos, Bertrand,Danascimento, Sophie,Meudal, Hervé,Noble, Florence,Garbay, Christiane,Roques, Bernard P.
, p. 3947 - 3956 (2007/10/03)
To improve our knowledge of the bioactive conformation of CCK-B antagonists, we have developed a new series of constrained dipeptoids whose synthesis and biochemical properties are reported here. These compounds, of general structure N(α)-[(2-adamantyloxy