203924-60-1Relevant articles and documents
Discovery and evaluation of pyrazolo[1,5-a]pyrimidines as neuropeptide Y1 receptor antagonists
Griffith, David A.,Hargrove, Diane M.,Maurer, Tristan S.,Blum, Charles A.,De Lombaert, Stéphane,Inthavongsay, John K.,Klade, Lee E.,MacK, Christine M.,Rose, Colin R.,Sanders, Martin J.,Carpino, Philip A.
scheme or table, p. 2641 - 2645 (2011/06/20)
A novel series of pyrazolo[1,5-a]pyrimidine derivatives was synthesized and evaluated as NPY Y1R antagonists. High binding affinity and selectivity were achieved with C3 trisubstituted aryl groups and C7 substituted 2-(tetrahydro-2H-pyran-4-ylamino)ethyla
SUBSTITUTED 6,5-HETERO-BICYCLIC DERIVATIVES
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, (2008/06/13)
This invention relates to compounds of the formula wherein A, B, D, E K, I, G, R3 and R5 are defined as in the specification, and to the pharmaceutically acceptable salts of such compounds.