212578-44-4Relevant articles and documents
Chromanylurea compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor and uses thereof
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Page/Page column 21, (2008/06/13)
Compounds that are antagonists of the VR1 receptor, having formula (I) [image] or a pharmaceutically acceptable salt, prodrug, or salt of a prodrug thereof, wherein A1, A2, A3, A4, R7, R8, R9, X, Y, Z, L, n, and m, are as defined herein, and are useful in disorders prevented or ameliorated by inhibiting the VR1 receptor.
New substituted 1,4-benzoxazine derivatives with potential intracellular calcium activity
Bourlot, Anne-Sophie,Sánchez, Isabel,Dureng, Georges,Guillaumet, Gérald,Massingham, Roy,Monteil, André,Winslow, Eileen,Pujol, M. Dolors,Mérour, Jean-Yves
, p. 3142 - 3158 (2007/10/03)
Substituted 1,4-benzoxazines bearing an amino side chain at the 2- position were prepared and were found to have a moderate activity on intracellular calcium. Of the compounds studied it was found that those which possess a homoveratrylamino moiety exhibi