226724-42-1Relevant articles and documents
Human beta3 adrenergic receptor agonists containing cyclic ureidobenzenesulfonamides.
Parmee,Naylor,Perkins,Colandrea,Ok,Candelore,Cascieri,Deng,Feeney,Forrest,Hom,MacIntyre,Miller,Stearns,Strader,Tota,Wyvratt,Fisher,Weber
, p. 749 - 754 (2007/10/03)
Human beta3 adrenergic receptor agonists containing 5-membered ring ureas were shown to be potent partial agonists with excellent selectivity over beta1 and beta2 binding. L-760,087 (4a) and L-764,646 (5a) (beta3 EC50 = 18 and 14 nM, respectively) stimula