24003-71-2Relevant articles and documents
GRANZYME B DIRECTED IMAGING AND THERAPY
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Page/Page column 82; 98, (2019/09/04)
Provided herein are heterocyclic compounds useful for imaging Granzyme B. Methods of imaging Granzyme B, combination therapies, and kits comprising the Granzyme B imaging agents are also provided.
Regioselective synthesis of tetrasubstituted pyrroles by 1,3-dipolar cycloaddition and spontaneous decarboxylation
Kim, Yongju,Kim, Jonghoon,Park, Seung Bum
supporting information; experimental part, p. 17 - 20 (2009/08/07)
We developed a novel regioselective synthesis of tetrasubstituted pyrroles via the classic 1,3-dipolar cycloaddition of α,β-unsaturated benzofuran-3(2H)-one and azlactones (1) followed by spontaneous decarboxylation. The complete regiochemical control of tetrasubstituted pyrroles was confirmed by the orthogonal synthesis of complementary regioisomers (7a and 7b) simply by using different azlactones (1a and 1b, respectively).
INTER VS INTRAMOLECULAR AMIDOALKYLATIONS OF AROMATICS - A NEW SYNTHESIS OF OXINDOLES, ISOQUINOLONES AND BENZAZEPINONES
Ben-Ishai, D.,Peled, N.,Sataty, I
, p. 569 - 572 (2007/10/02)
A new synthesis of oxindoles (8) isoquinolones (5) and benzazepinones (10) by the intramolecular amidoalkylation of aromatic amides of bismethoxycarbonylaminoacetic acid (4, 7, 9) is described.