255847-14-4Relevant articles and documents
Discovery of novel neuronal voltage-dependent calcium channel blockers based on emopamil left hand as a bioactive template
Suzuki, Yuichi,Yamamoto, Noboru,Iimura, Yoichi,Kawano, Koki,Kimura, Teiji,Nagato, Satoshi,Ito, Koichi,Komatsu, Makoto,Norimine, Yoshihiko,Kimura, Manami,Teramoto, Tetsuyuki,Kaneda, Yoshihisa,Hamano, Takeshi,Niidome, Tetsuhiro,Yonaga, Masahiro
, p. 919 - 922 (2007/10/03)
A series of novel neuronal voltage-dependent calcium channel (VDCC) blockers, with inhibitory activity at low micromolar and moderate solubility in water, was discovered by constructing and screening a focused library based on emopamil (1) left hand (ELH)