27464-01-3Relevant articles and documents
Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5- b]pyridazines for the Treatment of Human African Trypanosomiasis
Tear, Westley F.,Bag, Seema,Diaz-Gonzalez, Rosario,Ceballos-Pérez, Gloria,Rojas-Barros, Domingo I.,Cordon-Obras, Carlos,Pérez-Moreno, Guiomar,García-Hernández, Raquel,Martinez-Martinez, Maria Santos,Ruiz-Perez, Luis Miguel,Gamarro, Francisco,Gonzalez Pacanowska, Dolores,Caffrey, Conor R.,Ferrins, Lori,Manzano, Pilar,Navarro, Miguel,Pollastri, Michael P.
, p. 756 - 783 (2020/02/04)
From a high-throughput screen of 42 44 known human kinases inhibitors, a pyrazolo[1,5-b]pyridazine scaffold was identified to begin optimization for the treatment of human African trypanosomiasis. Previously reported data for analogous compounds against h
Synthesis of 3-hydrazino-pyridazines with basic substituents in 6 positions, with hypotensive activity
Bellasio,Parravicini,Testa
, p. 919 - 929 (2007/10/05)
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