32500-66-6Relevant articles and documents
Preliminary structure-activity relationship (SAR) of a novel series of pyrazole SKF-96365 analogues as potential store-operated calcium entry (SOCE) inhibitors
Dago, Camille D.,Le Maux, Paul,Roisnel, Thierry,Brigaudeau, Christophe,Bekro, Yves-Alain,Mignen, Olivier,Bazureau, Jean-Pierre
, (2018/03/25)
From a series of (1R, 1S)-1[β-(phenylalkoxy)-(phenetyl)]-1H-pyrazolium hydrochloride as new analogues of SKF-96365, one has an interesting effect for endoplasmic reticulum (ER) Ca2+ release and store-operated Ca2+ entry (SOCE) (ICsu
An efficient synthesis of β-hydroxyethylpyrazoles from propylene and styrene oxide using Cs2CO3
Duprez, Virginie,Heumann, Andreas
, p. 5697 - 5701 (2007/10/03)
Bases such as caesium carbonate efficiently catalyze the regioselective ring opening of propylene and styrene oxide with various substituted pyrazoles.
Effects of base, electrophile, and substrate on the selective alkylation of heteroaromatic systems
Smith, Thomas E.,Mourad, Michelle S.,Velander, Alan J.
, p. 1211 - 1217 (2007/10/03)
Several heteroaromatic systems, including oxazoles, pyrazoles, and thiophenes, are regioselectively alkylated using lithium diethylamide. Effects of substrate, base, and electrophile on the selectivity of this process are surveyed and interpreted.