3283-79-2Relevant articles and documents
Synthesis and Biological Evaluation of Novel Bischalcone Derivatives as Carbonic Anhydrase Inhibitors
Arslan, Tayfun,?elik, Gonca,?elik, Habip,?entürk, Murat,Yayl?, Nurettin,Ekinci, Deniz
, p. 741 - 748 (2016)
Design and synthesis of a new type of bischalcones as an alternative to natural and synthetic bischalcones are reported for the first time. Key steps involved the solvent-free Claisen–Schmidt condensation of chalcones, and the successful first application
Synthesis and bioactivity evaluation of eugenol hybrids obtained by Mannich and 1,3 dipolar cycloaddition reactions
Buduma, Komuraiah,Kumar A, Niranjana,Srinivas KVN, Satya,Kumar J, Kotesh,Chinde, Srinivas,Domatti, Anand Kumar,Kumar, Yogesh,Grover, Paramjit,Tiwari, Ashok,Khan, Feroz
, p. 2078 - 2089 (2021/07/10)
Design, synthesis, and bioactivity evaluation of novel mannich bases (2a-2j) and triazole-chalcone derivatives (7a-7k) of Eugenol 1 were reported. Among all the derivatives tested for antiproliferative activity, di-amine manich derivative 2b (32.92 μM), a
Synthesis and Pharmacological Investigations of Novel Pyrazolyl and Hydrazonoyl Cyanide Benzimidazole Entities
Khalifa, Mohamed E.,Gobouri, Adil A.,Kabli, Fahad M.,Altalhi, Tariq A.,Almalki, Abdulraheem S. A.,Elemshaty, Amira M.
, p. 1426 - 1436 (2019/04/17)
Various novel benzimidazole entities linked to pyrazolyl and hydrazonoyl cyanide substrates carrying aryl and heteroaryl groups (8a–e to 10a–e) were synthesized using new route syntheses and were focused on their pharmacological evaluation as one of the m
