329347-25-3Relevant articles and documents
Facile synthesis of 7-10 membered rings by intramolecular condensation using dialkylcarbonate as solvent
Ikemoto, Tomomi,Ito, Tatsuya,Nishiguchi, Atsuko,Tomimatsu, Kiminori
, p. 9335 - 9339 (2004)
A convenient large-scalable synthesis of 1-benzazepines 19 as an important intermediate of CCR5 antagonist, oral HIV-1 therapy, was established. The anilination of o-halogenobenzaldehyde 9 with alkylamino-acid 16 gave o-formylaniline-acid 17. Compound 17