343616-01-3Relevant articles and documents
An efficient synthesis of sulfamides
Guo, Chuangxing,Dong, Liming,Kephart, Susan,Hou, Xinjun
supporting information; experimental part, p. 2909 - 2913 (2010/06/14)
Here we report an efficient synthesis of sulfamides. 3,5-Lutidine was found to be an optimal solvent and catalyst for the reaction. The method was developed during our efforts to synthesize a series of novel FKBP-12 inhibitors in which the known ketoamide linker was replaced with sulfamide.