35973-84-3Relevant articles and documents
Novel compounds and their use in therapy
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Page/Page column 29, (2008/06/13)
Thiophenepyrimidinone compounds and their use in therapy, especially for use in the treatment and/or prevention of a steroid hormone dependent diseases or disorders, such as steroid hormone dependent diseases or disorders requiring inhibition of 17β-hydroxysteroid dehydrogenase enzymes.
Convenient Heterocyclization Reactions with Ethyl 2-Amino-4,5,6,7-tetrahydrobenzothiophene-3-carboxylate: Synthesis of Thiazole, Isoxazole, Pyrazole, Pyrimidine and Pyridazine Derivatives
Zohdi, Hussein F.,Wardakhan, Wagnat W.,Doss, Senot H.,Mohareb, Rafat M.
, p. 2526 - 2545 (2007/10/03)
Ethyl 2-amino-4,5,6,7-tetrahydrobenzothiophene-3-carboxylate (1) reacts with different reagents to afford thiazole, pyrazole, isoxazole, pyrimidine and pyridazine derivatives with interesting biological activities.
Synthesis of 2-methyl, 3-aryl or arylalkyl 5,6-dimethyl or Polymethylene Thieno -pyrimidine-4-ones
Kulshreshtha, M. J.,Bhatt, Shailendra,Pardasani, Madhuri,Khanna, N. M.
, p. 982 - 984 (2007/10/02)
Synthesis of 2-methyl, 3-aryl or arylalkyl 5,6-dimethyl or polymethylene thieno -pyrimidine-4-ones is described.A few compounds showed weak diuretic, hypotensive and anti-inflammatory activity.