3694-49-3Relevant articles and documents
Characterization of the binding site of the histamine H3 receptor. 2. Synthesis, in vitro pharmacology, and QSAR of a series of monosubstituted benzyl analogues of thioperamide
Windhorst, Albert D.,Timmerman, Henk,Worthington, Edward A.,Bijloo, Greetje J.,Nederkoorn, Paul H. J.,Menge, Wiro M. P. B.,Leurs, Rob,Herscheid, Jacobus D. M.
, p. 1754 - 1761 (2007/10/03)
A series of monosubstituted benzyl analogues of the histamine H3 receptor antagonist thioperamide were synthesized and evaluated for their histamine H3 receptor activity on the guinea pig jejunum. Incorporation of Cl, Br, and I at th