38912-41-3Relevant articles and documents
Antimicrobial activity of new benzazolyl N-sulfonyl amidines
Bakulev, Vasiliy A.,Beryozkina, Tetyana V.,Eltsov, Oleg S.,Fan, Zhijin,Galieva, Nadezhda A.,Lubec, Gert,Saveliev, Dmitriy A.,Xing, Jihong
, p. 495 - 497 (2021)
The reactions of N-(benz[d]oxazol-2-yl)- or N-(benzo[d]-thiazol-2-yl)-substituted carbothioamides with sulfonyl azides proceed as replacement of thioxo substituent by the sulfonylimino group to afford the corresponding N'-sulfonylated amidines. Acetic acid thioamides react smoothly upon boiling in ethanol, while for thioamides of trifluoroacetic and benzoic acids heating to 80–90 °C was required. Among hybrid molecules thus prepared, bacteriostatic-, bactericidal- and fungistatic-active against S. aureus and C. albicans representatives were found.
SPECTRAL INVESTIGATIONS OF THE TAUTOMERIC EQUILIBRIA OF THIOACYL DERIVATIVES OF 2-AMINOTHIAZOLE AND 2-AMINOBENZOTHIAZOLE
Jagodzinski, T.,Jagodzinska, E.,Dziembowska, T.,Szczodrowska, B.
, p. 337 - 344 (2007/10/02)
The positions of the tautomeric equilibria for a number of thioacyl derivatives of 2-aminothiazole and 2-aminobenzothiazole were determined by UV and IR spectroscopy with the use of model compounds.Quantum-chemical calculations by the CNDO/2 method were m
