40029-93-4Relevant articles and documents
Unexpected tandem condensation of 2-furonitriles with diethylenetriamine
Terenin,Galkin,Kabanova,Ivanov
, p. 351 - 353 (2010)
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Efficient synthesis of 2-imidazolines in the presence of molecular iodine under ultrasound irradiation
Chen, Guo-Feng,Li, Hong-Yang,Xiao, Nan,Chen, Bao-Hua,Song, Ya-Li,Li, Ji-Tai,Li, Zhi-Wei
, p. 1516 - 1521 (2014/12/11)
An efficient one-pot synthesis process for preparing 2-imidazolines from aldehydes and ethylenediamine using molecular iodine and potassium carbonate in absolute ethanol at 25-30°C under ultrasound irradiation is described. The synthetic strategy has the following advantages: mild conditions and low costs requirements, readily available catalyst, short reaction times, simplicity of operation, and good-to-excellent yields.
Novel diversely substituted 1-heteroaryl-2-imidazolines for fragment-based drug discovery
Krasavin, Mikhail
scheme or table, p. 2876 - 2880 (2012/07/28)
A palladium-catalyzed Buchwald-Hartwig arylation protocol has been applied to achieve high-yielding N-heteroarylation of a diverse set of privileged 2-imidazolines. The resulting compounds are of interest as a novel type of molecular tool for fragment-bas