409313-67-3Relevant articles and documents
[3-cis-3,5-dimethyl-(1-piperazinyl)alkyl]-bis-(4′-fluorophenyl)amine analogues as novel probes for the dopamine transporter
Cao, Jianjing,Husbands, Stephen M.,Kopajtic, Theresa,Katz, Jonathan L.,Newman, Amy Hauck
, p. 3169 - 3173 (2001)
In a continuing effort to identify novel probes with which to study the dopamine transporter (DAT), we discovered that the σ receptor antagonist, rimcazole, binds with moderate affinity (Ki=224 nM) to the DAT. The results from previous SAR stud